allosteric modulator
In pharmacology and biochemistry, allosteric modulators are a group of substances that bind to a Receptor (biochemistry), receptor to change that receptor's response to stimulus. Some of them, like benzodiazepines, are drugs. The site that an allos ...
of the
cannabinoid
Cannabinoids () are several structural classes of compounds found in the cannabis plant primarily and most animal organisms (although insects lack such receptors) or as synthetic compounds. The most notable cannabinoid is the phytocannabinoid tet ...
receptor
Receptor may refer to:
* Sensory receptor, in physiology, any structure which, on receiving environmental stimuli, produces an informative nerve impulse
*Receptor (biochemistry), in biochemistry, a protein molecule that receives and responds to a ...
.
See also
*
GAT100
GAT100 is a negative allosteric modulator of the cannabinoid CB1 receptor.
See also
* Org 27569
* PSNCBAM-1
* ZCZ-011
ZCZ-011 is a positive allosteric modulator of the cannabinoid
Cannabinoids () are several structural classes of co ...
*
Org 27569
Org 27569 is a drug which acts as a potent and selective negative allosteric modulator of the cannabinoid CB1 receptor. Studies ''in vitro'' suggest that it binds to a regulatory site on the CB1 receptor target, causing a conformational change t ...
*
ZCZ-011
ZCZ-011 is a positive allosteric modulator of the cannabinoid
Cannabinoids () are several structural classes of compounds found in the cannabis plant primarily and most animal organisms (although insects lack such receptors) or as synthetic c ...