WIN 54,461 (6-Bromopravadoline) is a drug that acts as a potent and selective
inverse agonist
In pharmacology, an inverse agonist is a drug that binds to the same receptor as an agonist but induces a pharmacological response opposite to that of the agonist.
A neutral antagonist has no activity in the absence of an agonist or inverse ago ...
for the
cannabinoid receptor
Cannabinoid receptors, located throughout the body, are part of the endocannabinoid system a class of cell membrane receptors in the G protein-coupled receptor superfamily. As is typical of G protein-coupled receptors, the cannabinoid recep ...
CB2.
See also
*
AM-630 (6-Iodopravadoline)
*
WIN 48,098 (Pravadoline)
*
WIN 55,212-2
WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure.
WIN 55,212-2 is a potent canna ...
References
Cannabinoids
Aminoalkylindoles
WIN compounds
Benzoylindoles
4-Morpholinyl compunds
Organobromides
{{cannabinoid-stub