Trepipam (
INN
Inns are generally establishments or buildings where travelers can seek lodging, and usually, food and drink. Inns are typically located in the country or along a highway; before the advent of motorized transportation they also provided accommo ...
) is a
dopamine receptor
Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through diffe ...
agonist of the
benzazepine
Benzazepines are heterocyclic chemical compounds consisting of a benzene ring fused to an azepine ring. Examples include:
File:Benazepril structure.svg, Benazepril
File:Fenoldopam.svg, Fenoldopam
File:GSK-189,254.svg, GSK-189,254
File:Ivabradine ...
group that was never marketed.
It acts specifically as an agonist of the
dopamine D1 receptor.
It is closed related
structurally
A structure is an arrangement and organization of interrelated elements in a material object or system, or the object or system so organized. Material structures include man-made objects such as buildings and machines and natural objects such as ...
to
fenoldopam
Fenoldopam mesylate (Corlopam) is a drug and synthetic benzazepine derivative which acts as a selective D1 receptor partial agonist. Fenoldopam is used as an antihypertensive agent. It was approved by the Food and Drug Administration (FDA) in ...
, a
peripherally acting selective D
1 receptor partial agonist which is used as an
antihypertensive agent.
References
1-Phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines
Abandoned drugs
Benzazepines
D1-receptor agonists
{{drug-stub