Nafadotride
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Nafadotride is a
dopamine antagonist A dopamine antagonist, also known as an anti-dopaminergic and a dopamine receptor antagonist (DRA), is a type of drug which blocks dopamine receptors by receptor antagonism. Most antipsychotics are dopamine antagonists, and as such they have ...
with reasonable selectivity for the D3 subtype (9.6 times selectivity for D3 over D2).Pilla M, Perachon S, Sautel F, Garrido F, Mann A, Wermuth CG, Schwartz JC, Everitt BJ, Sokoloff P. Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 agonist. ''Nature''. 1999;400:371–375.


References

Dopamine antagonists Pyrrolidines Carboxamides Nitriles Naphthol ethers {{nervous-system-drug-stub