Isamoltane (CGP-361A) is a drug used in

scientific research The scientific method is an empirical method for acquiring knowledge that has characterized the development of science since at least the 17th century (with notable practitioners in previous centuries; see the article history of scientific m ...

. It acts as an antagonist at the β-adrenergic, 5-HT_1A, and 5-HT_1B receptors. It has about five times the potency for the 5-HT_1B receptor (21 nmol/L) over the 5-HT_1A receptor (112 nmol/L). It has

anxiolytic An anxiolytic (; also antipanic or antianxiety agent) is a medication or other intervention that reduces anxiety. This effect is in contrast to anxiogenic agents which increase anxiety. Anxiolytic medications are used for the treatment of anxiet ...

effects in rodents.

References

{{Serotonin receptor modulators 5-HT1A antagonists 5-HT1B antagonists Secondary alcohols Beta blockers Phenol ethers Pyrroles Isopropyl compounds Amines