TRPM4-IN-5 is a drug which acts as a moderately potent but highly selective blocker of the

TRPM4 Transient receptor potential cation channel subfamily M member 4 (hTRPM4), also known as melastatin-4, is a protein that in humans is encoded by the TRPM4 gene. TRPM4 Channel Blocker * 9-Phenanthrol * TRPM4-IN-5 See also * TRPM TRPM is a family ...

ion channel, with an IC₅₀ of 1.5μM. It is protective against glutamate mediated neuronal excitotoxicity.

References

{{pharm-stub Carboxylic acids Amides Chlorobenzenes