Betamethadol (
INN
Inns are generally establishments or buildings where travelers can seek lodging, and usually, food and drink. Inns are typically located in the country or along a highway; before the advent of motorized transportation they also provided accommo ...
), or β-methadol, also known as betametadol, is a
synthetic opioid
Opioids are substances that act on opioid receptors to produce morphine-like effects. Medically they are primarily used for pain relief, including anesthesia. Other medical uses include suppression of diarrhea, replacement therapy for opioid us ...
analgesic
An analgesic drug, also called simply an analgesic (American English), analgaesic (British English), pain reliever, or painkiller, is any member of the group of drugs used to achieve relief from pain (that is, analgesia or pain management). It ...
.
It is an
isomer
In chemistry, isomers are molecules or polyatomic ions with identical molecular formulae – that is, same number of atoms of each element – but distinct arrangements of atoms in space. Isomerism is existence or possibility of isomers.
Iso ...
of
dimepheptanol
Dimepheptanol (International nonproprietary name, INN; Amidol, Pangerin), also known as methadol or racemethadol, is a Chemical synthesis, synthetic opioid analgesic related to methadone. It has similar effects to other opioids, including Analge ...
(methadol), the other being
alphamethadol
Alphamethadol ( INN), or α-methadol, also known as alfametadol, is a synthetic opioid analgesic. It is an isomer of dimepheptanol (methadol), the other being betamethadol (β-methadol). Alphamethadol is composed of two isomers itself, L-α-met ...
(α-methadol).
Betamethadol is composed of two isomers itself,
L-β-methadol, and
D-β-methadol.
Based on
structure-activity relationships it can be inferred that both isomers are likely to be
active
Active may refer to:
Music
* ''Active'' (album), a 1992 album by Casiopea
* Active Records, a record label
Ships
* ''Active'' (ship), several commercial ships by that name
* HMS ''Active'', the name of various ships of the British Royal ...
as opioid analgesics, similarly to those of
betacetylmethadol
Betacetylmethadol is a Chemical synthesis, synthetic opioid. It is a diastereoisomer of alphacetylmethadol (as well as levacetylmethadol). In the United States, betacetylmethadol is a List of Schedule I drugs (US), Schedule I drug Narcotic under ...
(β-acetylmethadol).
See also
*
Dimepheptanol
Dimepheptanol (International nonproprietary name, INN; Amidol, Pangerin), also known as methadol or racemethadol, is a Chemical synthesis, synthetic opioid analgesic related to methadone. It has similar effects to other opioids, including Analge ...
*
Alphamethadol
Alphamethadol ( INN), or α-methadol, also known as alfametadol, is a synthetic opioid analgesic. It is an isomer of dimepheptanol (methadol), the other being betamethadol (β-methadol). Alphamethadol is composed of two isomers itself, L-α-met ...
*
Betacetylmethadol
Betacetylmethadol is a Chemical synthesis, synthetic opioid. It is a diastereoisomer of alphacetylmethadol (as well as levacetylmethadol). In the United States, betacetylmethadol is a List of Schedule I drugs (US), Schedule I drug Narcotic under ...
References
Secondary alcohols
Dimethylamino compounds
Analgesics
Mu-opioid receptor agonists
Synthetic opioids
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